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PK Parameter Database

83 drugs — t½, Vd, CL, F, PPB, MW. Click any row for full detail and source.

83 drugs
Drug Class t½ (h) Vd (L/kg) F (%) PPB (%) MW
AmitriptylineTricyclic antidepressant21.015.04895.0277
AmlodipineCalcium channel blocker (DHP)40.021.06493.0409
AmoxicillinAminopenicillin1.100.269318.0365
ApixabanDirect oral anticoagulant (FXa inhibitor)12.00.535087.0460
Aspirin (Acetylsalicylic acid)NSAID / Antiplatelet0.250.156880.0180
Atenololβ₁-blocker6.500.67505.00266
AtorvastatinStatin (HMG-CoA reductase inhibitor)14.05.801498.0559
AzithromycinMacrolide antibiotic68.031.03751.0749
Bisoprololβ₁-blocker11.03.509030.0325
CaffeineMethylxanthine / CNS stimulant4.500.6110036.0194
CarbamazepineAnticonvulsant / Mood stabiliser15.01.407875.0236
CelecoxibNSAID (COX-2 selective)11.06.009997.0381
CetirizineAntihistamine (H₁, non-sedating)7.500.507093.0389
Ciclosporin (Cyclosporine)Calcineurin inhibitor8.403.503098.01,202.6
CiprofloxacinFluoroquinolone antibiotic4.502.507030.0331
ClindamycinLincosamide antibiotic2.501.109094.0425
ClopidogrelAntiplatelet (P2Y12 inhibitor)7.500.505098.0322
CodeineOpioid3.003.60537.00299
DexamethasoneCorticosteroid4.000.827877.0393
DiazepamBenzodiazepine43.01.1010099.0285
DiclofenacNSAID1.100.175499.0296
DigoxinCardiac glycoside36.07.307525.0781
DoxycyclineTetracycline antibiotic18.00.759390.0444
EscitalopramSSRI27.012.08056.0324
EthanolAlcohol0.250.60800.0046.1
EthinylestradiolSynthetic oestrogen13.04.304598.0296
FentanylOpioid (short-acting IV)3.504.003284.0337
FluoxetineSSRI53.035.07294.0309
FurosemideLoop diuretic1.500.115299.0331
GabapentinAnticonvulsant / Neuropathic pain6.000.65600.00171
GentamicinAminoglycoside antibiotic2.500.26010.0478
Glibenclamide (Glyburide)Sulfonylurea (antidiabetic)10.00.139999.0494
HaloperidolAntipsychotic (typical, D₂ antagonist)21.018.06092.0376
HydroxychloroquineAntimalarial / DMARD1,3447507450.0336
IbuprofenNSAID2.000.158099.0206
ImatinibTyrosine kinase inhibitor (BCR-ABL)18.04.909895.0494
KetamineDissociative anaesthetic / NMDA antagonist2.503.102047.0238
LamotrigineAnticonvulsant / Mood stabiliser29.01.109855.0256
LevetiracetamAnticonvulsant (SV2A)7.000.591000.00170
Levothyroxine (T4)Thyroid hormone1680.138099.0799
LisinoprilACE inhibitor12.00.75250.00442
LithiumMood stabiliser22.00.791000.006.90
LoperamideAntidiarrhoeal (peripheral µ-opioid)11.02.804097.0477
LoratadineAntihistamine (H₁, non-sedating)8.401195397.0383
LorazepamBenzodiazepine14.01.309391.0321
MelatoninPineal hormone / Chronobiotic0.750.821560.0232
MetforminBiguanide (antidiabetic)4.503.70500.00166
MethotrexateAntimetabolite / DMARD10.00.557050.0454
Metoprololβ₁-blocker3.504.003812.0267
MetronidazoleNitroimidazole antibiotic8.500.749920.0171
MidazolamBenzodiazepine2.501.104497.0326
MontelukastLeukotriene receptor antagonist4.500.156499.0586
MorphineOpioid2.503.502435.0285
NaloxoneOpioid antagonist1.102.60245.0327
NaproxenNSAID14.00.169999.0230
NicotinenAChR agonist / Alkaloid2.002.60115.00162
NitrofurantoinNitrofuran antibiotic0.500.778760.0238
OlanzapineAntipsychotic (atypical)33.016.05793.0312
OmeprazoleProton pump inhibitor1.000.345297.0345
Ondansetron5-HT₃ antagonist (antiemetic)3.501.906073.0293
OseltamivirNeuraminidase inhibitor (antiviral)1.500.357542.0312
PantoprazoleProton pump inhibitor1.200.157798.0383
Paracetamol (Acetaminophen)Analgesic2.200.908520.0151
PhenytoinAnticonvulsant (Na⁺ channel)22.00.649090.0252
PrednisoloneCorticosteroid3.500.518270.0360
PropofolIV anaesthetic agent5.004.00098.0178
QuetiapineAntipsychotic (atypical)7.0010.0983.0384
RamiprilACE inhibitor13.01.202873.0417
Salbutamol (Albuterol)β₂-agonist SABA3.800.47118.00239
SertralineSSRI26.020.04498.0306
SildenafilPDE5 inhibitor4.001.704196.0475
SimvastatinStatin (HMG-CoA reductase inhibitor)2.505.00595.0419
SpironolactonePotassium-sparing diuretic (aldosterone antagonist)1.600.056598.0417
TacrolimusCalcineurin inhibitor12.01.902599.0804
TamoxifenSERM (selective oestrogen receptor modulator)16850.09999.0372
Tenofovir disoproxil fumarateNRTI (antiretroviral)17.01.30257.00287
TheophyllineXanthine bronchodilator9.000.489656.0180
TramadolOpioid (atypical)6.002.707520.0263
Valproate (Valproic acid)Anticonvulsant / Mood stabiliser14.00.2210093.0166
VancomycinGlycopeptide antibiotic6.000.70055.01,449.3
VenlafaxineSNRI5.007.504527.0277
VerapamilCalcium channel blocker (non-DHP)6.505.502290.0455
WarfarinVitamin K antagonist40.00.149999.0308

Values are typical population averages for healthy adults from Rowland & Tozer Clinical Pharmacokinetics (5th ed.), Brunton et al. Goodman & Gilman's (13th ed.), and Bauer Clinical Pharmacokinetics Handbook (2nd ed.). Click any row for individual source citation and full parameter detail.